2012年1月
Synthesis of (-)-benzolactam-V8 by application of asymmetric aziridination
TETRAHEDRON
- ,
- ,
- ,
- ,
- 巻
- 68
- 号
- 3
- 開始ページ
- 878
- 終了ページ
- 882
- 記述言語
- 英語
- 掲載種別
- 研究論文(学術雑誌)
- DOI
- 10.1016/j.tet.2011.11.033
- 出版者・発行元
- PERGAMON-ELSEVIER SCIENCE LTD
(-)-Benzolactam-V8, an artificially-designed cyclic dipeptide with strong tumor-promoter activity, was synthesized from benzyl (S)-N-(2-formylphenyl)-N-methylvalinate by application of guanidinium ylideparticipated asymmetric aziridination followed by the reductive ring-opening reaction of 3-arylaziridine-2-carboxylate formed. (C) 2011 Elsevier Ltd. All rights reserved.
- リンク情報
- ID情報
-
- DOI : 10.1016/j.tet.2011.11.033
- ISSN : 0040-4020
- Web of Science ID : WOS:000299609300012