佐々木秀 (Shigeru Sasaki) - マイポータル

基本情報

所属: 星薬科大学医薬品化学研究所有機合成化学研究室助教

学位: 博士（薬学）(2014年3月星薬科大学)

J-GLOBAL ID: 201601013774142370
researchmap会員ID: B000252097

研究分野

ライフサイエンス / 薬系化学、創薬科学 /

論文

Further investigation of the rapid-onset and short-duration action of the G protein-biased μ-ligand oliceridine

Tomohisa Mori, Yoshinori Takemura, Takamichi Arima, Yoshiyuki Iwase, Michiko Narita, Kanako Miyano, Yusuke Hamada, Yukari Suda, Akinobu Matsuzawa, Kazuyuki Sugita …

Biochemical and Biophysical Research Communications 534 988-994 2021年1月1日
Transition-Metal-Free Synthesis of Pyridine Derivatives by Thermal Cyclization of N -Propargyl Enamines

Yuya Chikayuki, Takakane Miyashige, Shiori Yonekawa, Akiko Kirita, Natsuko Matsuo, Hiroyoshi Teramoto, Shigeru Sasaki, Kimio Higashiyama, Takayasu Yamauchi

Synthesis (Germany) 52(7) 1113-1121 2020年4月査読有り
Transition metal-free cyclization of N-boc-N-propargylenamines

Yuya Chikayuki, Yasuaki Kouno, Shiori Yonekawa, Haruka Ishikawa, Yoko Waki, Hiroyoshi Teramoto, Shigeru Sasaki, Kimio Higashiyama, Takayasu Yamauchi

Heterocycles 100(5) 719-746 2020年査読有り
Synthesis of thiourea derivatives from m-methoxycinnamic acid as antiangiogenic candidate

Juni Ekowati, Iwan Sahrial Hamid, Kholis Amalia Nofianti, Shigeru Sasaki

Jurnal Teknologi 81(4) 105-114 2019年査読有り
Substituent effects in regio- And stereoselective ring-opening reaction of aziridines with ET3N·3HF for β-fluoroamine synthesis

Shigeru Sasaki, Satono Watanabe, Kaori Shiino, Yuko Yanaka, Shiho Kaneko, Kana Miyamoto, Ayano Yasui, Hina Sakaino, Hiroyoshi Teramoto, Takayasu Yamauchi …

Heterocycles 97(2) 823-841 2018年査読有り
Synthesis of α,α-difluoro-β-hydroxy ketone via the La(OTf)<inf>3</inf>-catalyzed aldol reaction of carbonyl compounds with difluoroenol O-Boc esters

Shigeru Sasaki, Tatuo Suzuki, Toshihiro Uchiya, Shigenobu Toyota, Akira Hirano, Mao Tanemura, Hiroyoshi Teramoto, Takayasu Yamauchi, Kimio Higashiyama

Journal of Fluorine Chemistry 192 78-85 2016年査読有り
Design and synthesis of a piperidinone scaffold as an analgesic through kappa-opioid receptor: Structure-activity relationship study of matrine alkaloids

Hiroyoshi Teramoto, Takayasu Yamauchi, Yasushi Terado, Sanae Odagiri, Shigeru Sasaki, Kimio Higashiyama

Chemical and Pharmaceutical Bulletin 64(5) 410-419 2016年査読有り
Development of κ opioid receptor agonists by focusing on phenyl substituents of 4-dimethylamino-3-phenylpiperidine derivatives: Structure-activity relationship study of matrine type alkaloids

Hiroyoshi Teramoto, Takayasu Yamauchi, Shigeru Sasaki, Kimio Higashiyama

Chemical and Pharmaceutical Bulletin 64(5) 420-431 2016年査読有り
Bisoxazoline-catalyzed asymmetric nucleophilic addition of diethyl zinc to fluorinated alkyl ketones: Enantiofacial control by changing the bisoxazoline substituent

Shigeru Sasaki, Takayasu Yamauchi, Masatomi Kanai, Akihiro Ishii, Kimio Higashiyama

Bulletin of the Chemical Society of Japan 88(1) 200-208 2015年査読有り
Total synthesis of the proposed structures of eushearilide

Takayasu Yamauchi, Jun Ichi Takidaira, Kenya Okamoto, Takaya Sugiura, Hiroki Horikoshi, Shintaro Kudo, Shigeru Sasaki, Noriko Mizushima, Kimio Higashiyama

Heterocycles 88(2) 1175-1189 2014年査読有り
Structure modification of ethyl p-methoxycinnamate and their bioassay as chemopreventive agent against mice's fibrosarcoma

Juni Ekowati, Bimo A. Tejo, Shigeru Sasaki, Kimio Highasiyama, Sukardiman, Siswandono, Tutuk Budiati

International Journal of Pharmacy and Pharmaceutical Sciences 4(SUPPL.3) 528-532 2012年査読有り
Brønsted acid catalyzed friedel-crafts alkylation reactions of trifluoromethyl-α,β-ynones with indoles

Shigeru Sasaki, Yuta Ikekame, Manabu Tanayama, Takayasu Yamauchi, Kimio Higashiyama

Synlett 23(18) 2699-2703 2012年査読有り
Direct aldol reaction of trifluoromethyl ketones with ketones catalyzed by Et<inf>2</inf>Zn and secondary amines

Shigeru Sasaki, Kasumi Kikuchi, Takayasu Yamauchi, Kimio Higashiyama

Synlett (10) 1431-1434 2011年査読有り
Efficient microwave-assisted prenylation of pinostrobin and biological evaluation of its derivatives as antitumor agents

Hadi Poerwono, Shigeru Sasaki, Yoshiyuki Hattori, Kimio Higashiyama

Bioorganic and Medicinal Chemistry Letters 20(7) 2086-2089 2010年4月査読有り
Dy(OTf)3/Pybox-catalyzed enantioselective Friedel-Crafts alkylation of indoles with α,β-unsaturated trifluoromethyl ketones

Shigeru Sasaki, Takayasu Yamauchi, Kimio Higashiyama

Tetrahedron Letters 51(17) 2326-2328 2010年4月査読有り
Chemoselective reduction of ketones: Trifluoromethylketones versus methylketones

Shigeru Sasaki, Takayasu Yamauchi, Hajime Kubo, Masatomi Kanai, Akihiro Ishii, Kimio Higashiyama

Tetrahedron Letters 46(9) 1497-1500 2005年2月28日査読有り

共同研究・競争的資金等の研究課題

抗体薬物複合体における糖鎖構造の役割の解明と高機能化

日本学術振興会科学研究費助成事業基盤研究(B) 2019年4月 - 2023年3月

眞鍋史乃, 安永正浩, 松村保広, 羽場宏光, 佐々木秀

佐々木秀

基本情報

研究分野

論文

共同研究・競争的資金等の研究課題

メニュー

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