Aug, 2013
Chiral Phosphoric Acid-Catalyzed Oxidative Kinetic Resolution of Indolines Based on Transfer Hydrogenation to Imines
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
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- ,
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- Volume
- 135
- Number
- 32
- First page
- 11740
- Last page
- 11743
- Language
- English
- Publishing type
- Research paper (scientific journal)
- DOI
- 10.1021/ja406004q
- Publisher
- AMER CHEMICAL SOC
The oxidative kinetic resolution of 2-substituted indoline derivatives was achieved by hydrogen transfer to imines by means of a chiral phosphoric acid catalyst. The oxidative kinetic resolution was applicable to racemic alkyl- or aryl-substituted indolines, and the remaining indolines were obtained in good yields with excellent enantioselectivities.
- Link information
- ID information
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- DOI : 10.1021/ja406004q
- ISSN : 0002-7863
- Web of Science ID : WOS:000323241200016