間瀬年康 (Toshiyasu Mase) - マイポータル

A Scalable Process for the Synthesis of 2-Methyl-1,4,5,6- tetrahydroimidazo[4,5-d][1]benzazepine Monohydrate and 4-[(Biphenyl-2-ylcarbonyl)amino]benzoic Acid: Two New Key Intermediates for the Synthesis of the AVP Antagonist Conivaptan H・・・

Tsunoda, Takashi, Yamazaki, Atsuki, Mase, Toshiyasu, Sakamoto, Shuichi

Organic Process Research & Development 9(5) 593-598 2005年9月

A scalable process for the synthesis of 2-methyl-1,4,5,6-tetrahydroimidazo[4,5-d][1]benzazepine monohydrate and 4-[(biphenyl-2-ylcarbonyl)amino]benzoic acid: Two new key intermediates for the synthesis of the AVP antagonist conivaptan hydrochloride

T Tsunoda, A Yamazaki, T Mase, S Sakamoto

ORGANIC PROCESS RESEARCH & DEVELOPMENT 9(5) 593-598 2005年9月

A new synthetic route to YM087, an arginine vasopressin antagonist

T Tsunoda, A Tanaka, T Mase, S Sakamoto

HETEROCYCLES 63(5) 1113-1122 2004年5月

New thiazole derivatives as potent and selective 5-hydroxytriptamine 3 (5-HT3) receptor agonists for the treatment of constipation

Naoki Imanishi, Kiyoshi Iwaoka, Hiroyuki Koshio, Shin-Ya Nagashima, Ken-Ichi Kazuta, Mitsuaki Ohta, Shuichi Sakamoto, Hiroyuki Ito, Shinobu Akuzawa, Tetsuo Kiso …

Bioorganic and Medicinal Chemistry 11(7) 1493-1502 2003年4月

NMR structure of human fibronectin EDA

Niimi T, Osawa M, Yamaji N, Yasunaga K, Sakashita H, Mase T, Tanaka A, Fujita

J. of Biomolecular NMR, 21(3), 281-284(2001) 21(3) 281-264 2001年3月

NMR structure of human fibronectin EDA

J. of Biomolecular NMR, 21(3), 281-284(2001) 21(3) 281-264 2001年3月

A Novel Class of Inhibitors for Human Steroid 5α-Reductase: Synthesis and Biological Evaluation of Indoline and Aniline Derivatives. III

Igarashi S, Inami H, Hara H, Koutoku H, Oritani H, Mase T

Chem.Pharm.Bull.,48(11)1689-1697(2000) 48(11) 1689-1697 2000年11月

A Novel Class of Inhibitors for Human Steroid 5alalpha-Reductase: Synthesis and Biological Evaluation of Indoline and Aniline Derivatives. III

Susumu IGARASHI, Hiroshi INAMI, Hiromu HARA, Hiroshi KOUTOKU, Hiroyuki ORITANI, Toshiyasu MASE

Chem.Pharm.Bull.,48(11)1689-1697(2000) 48(11) 1689-1697 2000年11月

A Novel Class of Inhibitors for Human Steroid 5α-Reductase: Synthesis and Biological Evaluation of Indole Derivatives. II

Igarashi S, Inami H, Hara H, Fujii M, Koutoku H, Oritani H, Mase T

Chem.Pharm.Bull. 48(3) 382-388 2000年3月

A novel class of inhibitors for human steroid 5 alpha-reductase: Synthesis and biological evaluation of indole derivatives. II

S Igarashi, H Inami, H Hara, M Fujii, H Koutoku, H Oritani, T Mase

CHEMICAL & PHARMACEUTICAL BULLETIN 48(3) 382-388 2000年3月

A Novel Class of Inhibitors for Human Steroid 5α-Reductase: Phenoxybenzoic Acid Derivatives. I

Igarashi S, Kimura T, Naito R, Hara H, Fujii M, Koutoku H, Oritani H, Mase T

Chem.Pharm.Bull. 47(8) 1073-1080 1999年8月

A novel class of inhibitors for human steroid 5 alpha-reductase: Phenoxybenzoic acid derivatives. I

S Igarashi, T Kimura, R Naito, H Hara, M Fujii, H Koutoku, H Oritani, T Mase

CHEMICAL & PHARMACEUTICAL BULLETIN 47(8) 1073-1080 1999年8月

2-(3-Pyridyl)thiazolidine-4-carboxamide Derivatives.III. Synthesis of Metabolites and Metabolism of 2-(3-pyridyl)thiazolidine-4-carboxamides YM461 and YM264 as Platelet-Activating Factor(PAF) Receptor Antagonists

Suzuki T, Nagaoka H, Hara H, Takeuchi M, Saito M, Yamada T, Tomioka K, Matsumoto H, Takanuki K, Mase T

Chem. Pharm. Bull. 47(2) 165-170 1999年2月

2-(3-Pyridyl)thiazolidine-4-carboxamide Derivatives. III Synthesis of Metabolites and Metabolism of 2-(3-pyridyl)thiazolidine-4-carboxamides YM461 and YM264 as Platelet-Activating Factor(PAF) Receptor Antagonists

Takeshi SUZUKI, Hitoshi NAGAOKA, Hiromu HARA, Makoto TAKEUCHI, Munetoshi SAITO, Toshimitsu YAMADA, Kenichi TOMIOKA, Hisao MATSUMOTO, Kenichi TAKANUKI, Toshiyasu MASE

Chem. Pharm. Bull. 47(2) 165-170 1999年2月

Synthesis of the Selective 5-Hydroxytryptamine 4(5-HT4) Receptor Agonist (+)-(S)-2- Chloro-5-methoxy-4-[5-(2-piperidylmethyl)-1,2,4-oxazol-3-yl]aniline

Suzuki T, Iwaoka K, Imanishi N, Nagakura Y, Miyata K, Nakahara H, Ohta M, Mase T

Chem. Pharm. Bull 47(1) 120-122 1999年1月

Synthesis of the Selective 5-Hydroxytryptamine 4(5-HT4) Receptor Agonist (+)-(S)-2- Chloro-5-methoxy-4-[5-(2-piperidylmethyl)-1,2,4-oxazol-3-yl]aniline

Takeshi SUZUKI, Kiyoshi IWAOKA, Naoki IMANISHI, Yukinori NAGAKURA, Kenji MIYATA, Hideaki NAKAHARA, Mitsuaki OHTA, Toshiyasu MASE

Chem. Pharm. Bull 47(1) 120-122 1999年1月

2-(3-Pyridyl)thiazolidine-4-carboxamide Derivatives. Ⅱ. Structure-Activity Relationships and Active Configuration of 2-(3-Pyridyl)thiazolidine-4-carboxamides as Platelet-Activating Factor Receptor Antagonists

Suzuki T, Nagaoka H, Kondo Y, Takahashi T, Takeuchi M, Hara H, Saito M, Yamada T, Tomioka K, Hamada M …

Chem. Pharm. Bull. 46(9) 1468-1473 1998年9月

2-(3-Pyridyl)thiazolidine-4-carboxamide Derivatives.II. Structure-Activity Relationships and Active Configuration of 2-(3-Pyridyl)thiazolidine-4-carboxamides as Platelet-Activating Factor Receptor Antagonists

Takeshi SUZUKI, Hitoshi NAGAOKA, Yutaka KONDO, Takumi TAKAHASHI, Makoto TAKEUCHI, Hiromu HARA, Munetoshi SAITO, Toshimitsu YAMADA, Kenichi TOMIOKA, Mamoru HAMADA …

Chem. Pharm. Bull. 46(9) 1468-1473 1998年9月

Synthesis and pharmacological characterization of novel 6-fluorochroman derivatives as potential 5-HT(1A) receptor antagonists

Tomoyuki Yasunaga, Takenori Kimura, Ryo Naito, Toru Kontani, Fumikazu Wanibuchi, Hiroshi Yamashita, Tamako Nomura, Shin-Ichi Tsukamoto, Tokio Yamaguchi, Toshiyasu Mase

Journal of Medicinal Chemistry 41(15) 2765-2778 1998年7月16日

Novel 5-Hydroxytryptamine 4(5-HT4) Receptor Agonists. Synthesis and Gastroprokinetic Activity of 4-Amino-N-[2-(1-aminocycloalkan-1-yl)ethyl]-] 5-chloro-2-methoxybennzamides

Suzuki T, Imanishi N, Itahana H, Watanuki S, Miyata K, Ohta M, Nakahara H, Yamagiwa Y, Mase T

Chem. Pharm. Bull. 46(7) 1116-1124 1998年7月

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