論文

2022年

Discovery of a phase-separating small molecule that selectively sequesters tubulin in cells

Chemical Science
  • Genyir Ado
  • Naotaka Noda
  • Hue T. Vu
  • Amelie Perron
  • Amarjyoti D. Mahapatra
  • Karla Pineda Arista
  • Hideaki Yoshimura
  • Daniel M. Packwood
  • Fumiyoshi Ishidate
  • Shin-ichi Sato
  • Takeaki Ozawa
  • Motonari Uesugi
  • 全て表示

13
19
開始ページ
5760
終了ページ
5766
記述言語
掲載種別
研究論文(学術雑誌)
DOI
10.1039/d1sc07151c
出版者・発行元
Royal Society of Chemistry (RSC)

A non-peptidic small molecule, R-huezole, phase separates to selectively sequester tubulin proteins to control the cell cycle. Its modular structure provides a framework for designing bioactive molecules to mimic membraneless organelles in cells.

リンク情報
DOI
https://doi.org/10.1039/d1sc07151c
URL
http://pubs.rsc.org/en/content/articlepdf/2022/SC/D1SC07151C
ID情報
  • DOI : 10.1039/d1sc07151c
  • ISSN : 2041-6520
  • eISSN : 2041-6539

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